Retatrutide gaw, GLP-1, GIP, hte GCGRs ni hpe n-gun jaw na matu, GIP peptide backbone kaw na hkrang shapraw da ai amino acid 39 lawm ai peptide langai sha re.
Dai gaw, n-gun n rawng ai glucagon hormone receptor agonist (GLP-1, GIP, hte GCGR receptor ni) rai nna, 17.5% jan n-gun shayawm ai lam hpe lu la na matu, sai chyup ana n kap ai masha kaba ni hpe n-gun shayawm ya lu ai hpe mu lu ai, raitim, phase 2 chyam dinglik ai aten hta, n-gun ja ai (sh) n-gun ja ai (grai n-gun ja ai) ni hpe hkam la lu ai. Ndai chyam dinglik ai hta, tsi mawan law dik lu ai shanglawm ai ni gaw, bat 48 na ai hpang, 24.2% daram n-gun shayawm ai lam hpe madun dan ai.
Retatrutide gaw glucagon hkam la ai ni hpe madung tawn ai npawt nhpang triple agonist langai rai nna, glucagon hpe pat shingdang ai polypeptide, hte glucagon- zawn re ai peptide-1 hpe madung tawn ai. Retatrutide a yak hkak ai ladat gaw ndai hkam la ai ni a lapran hta synergistic matut mahkai lam lawm ai majaw, insulin hpe grau nna garan ginhka ai lam law wa ai, glucose homeostasis hpe grau kaja hkra galaw ya lu ai, n-gun ja ai malu masha hpe gram lajang lu ai. 1 kaw nna 3 du hkra na tsi rung chyam dinglik ai lam ni gaw, hkum hkrang n-gun hpe grai shayawm ya ai hte glycemic control mahtai ni hpe grai shayawm ya ai hku nna, ahkyak ai akyu rawng ai lam hpe madun dan sai. Dai hta n-ga, retatrutide gaw myit masin hte seng ai hkrit tsang hpa lam ni hpe shayawm ya lu ai hte metabolic n-gun n-gun yawm ai lam hpe hparan ai hta ga sadi jaw da ai-}associated steatotic ana zinli hpe tsun dan ai. Raitim, shi a aten galu shimlam masa hpe masat da na matu, laksan masha jahpan ni hta shi a atsam marai hpe sawk sagawn na matu, shi a karum shingtau ai tsi ladat ni hpe hpaw shadan dan na matu, ma ni a hpung ni hta shi a ladat ni hpe asan sha chye na hkra, atsawm sha myit maju jung ra ai. Galai shai wa ai tsi ladat langai hku nna, retatrutide gaw myit mada shara a beacon hpe madi madun ai, hkum hkrang n-gun ja ai hte 2 lang na hka n-gun n-rawng ai (T2DM) a hparan hpareng ai lam hta galai shai wa ai galai shai lam ni hpe madi madun ai, tsi gawk hta matut nna sawk sagawn ai lam hte gram lajang ai lam ni hpe galaw ra ai. Ndai labau hpe bai maram yu ai shaloi, hkum hkrang n-gun n-gun hte T2DM hpe hparan ai hta retatrutide a tsi ladat hpe sawk sagawn ai.
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